Written by Pitsinos M.
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Monday, 04 May 2009 12:56 |
- 1,1-Bis(phenylsulfonyl)-4-diethylamino-1,3-butadiene, a fully delocalized “push-pull” diene
Alcock, N.W.; Pike, G.A.; Papadopoulos, M.; Pitsinos, E.; Hatjiarapoglou, L.; Varvoglis, A. Phosphorus, Sulfur and Silicon and the Related Elements 1991, 60, 131–133
- Enantioselective total synthesis of (–)-calicheamicinone
Smith, A.L.; Hwang, C.-K.; Pitsinos, E.; Scarlato, G.R.; Nicolaou, K.C. Journal of the American Chemical Society 1992, 114, 3134–3136
- Total synthesis of calicheamicin gamma 1I
Nicolaou, K.C.; Hummel, C.W.; Pitsinos, E.N.; Nakada, M.; Smith, A.L.; Shibayama, K.; Saimoto, H. Journal of the American Chemical Society 1992, 114, 10082–10084
- Total synthesis of calicheamicin gamma 1I. 2. Development of an enantioselective route to (–)-calicheamicinone
Smith, A.L.; Pitsinos, E.N.; Hwang, C.-K.; Mizuno, Y.; Saimoto, H.; Scarlato, G.R.; Suzuki, T.; Nicolaou, K.C. Journal of the American Chemical Society 1993, 115, 7612–7624
- Total synthesis of calicheamicin gamma 1I. 3. The final stages
Nicolaou, K.C.; Hummel, C.W.; Nakada, M.; Shibayama, K.; Pitsinos, E.N.; Saimoto, H.; Mizuno, Y.; Baldenius, K.U.; Smith, A.L. Journal of the American Chemical Society 1993, 115, 7625–7635
- Synthetic calicheamicin mimics with novel initiation mechanisms: DNA cleavage, cytotoxicity, and apoptosis
Nicolaou, K.C.; Pitsinos, E.N.; Theodorakis, E.A.; Saimoto, H.; Wrasidlo, W. Chemistry & Biology 1994, 1, 57–66
- A water-soluble prodrug of Taxol with self-assembling properties
Nicolaou, K.C.; Guy, R.K.; Pitsinos, E.N.; Wrasidlo, W. Angewandte Chemie - International Edition in English 1994, 33, 1583–1587
- Inhibition of topoisomerase I by naphthoquinone derivatives
Papageorgiou, V. P.; Li T.; Plyta, Z. F.; Mellidis, A. S.; Assimopoulou, A. N.; Pitsinos, E. N.; Couladouros, E. A. Bioorganic and Medicinal Chemistry Letters 1998, 8, 3385–3390
- Stabilization of microtubules by combretastatin D derivatives
Couladouros, E. A.; Li, T.; Moutsos, V. I.; Pitsinos, E. N.; Soufli, I. C. Bioorganic and Medicinal Chemistry Letters 1999, 9, 2927–2928
- Biomimetic explorations towards the bisorbicillinoids. Total synthesis of bisorbicillinol, bisorbibutenolide and trichodimerol
Nicolaou, K. C.; Simonsen, K. B.; Vassilikogiannakis, G.; Baran, P. S.; Vidali, V. P.; Pitsinos, E. N.; Couladouros, E. A. Angewandte Chemie - International Edition 1999, 38, 3555–3559
- Biomimetic total synthesis of bisorbicillinol, bisorbibutenolide, trichodimerol, and designed analogues of bisorbicillinoids
Nicolaou, K. C.; Vassilikogiannakis, G.; Simonsen, K. B.; Baran, P. S.; Zhong, Y.-L.; Vidali, V. P.; Pitsinos, E. N.; Couladouros, E. A. Journal of the American Chemical Society 2000, 122, 3071–3079
- Vicinal tetraamines of defined geometry: Potential scaffolds for assembly
Pitsinos, E.N.; Lehn, J.-M.; De Cian, A. Helvetica Chimica Acta 2001, 84, 22–31
- Heterofunctional linking agents for the synthesis of well-defined block copolymers of dimethylsiloxane and tert-butyl methacrylate or 2-vinylpyridine
Bellas, V.; Iatrou, H.; Pitsinos, E.N.; Hadjichristidis, N. Macromolecules 2001, 34, 5376–5378
- A convenient route to alkaloid lipids: Application for the synthesis of a leptophylline A analogue
Koulocheri, S.D.; Pitsinos, E.N.; Haroutounian, S.A. Synthesis 2002, 111–115
- An expedient asymmetric synthesis of a calystegin B4 analogue
Koulocheri, S.D.; Pitsinos, E.N.; Haroutounian, S.A. Synthesis 2002, 1707–1710
- A novel 2΄-(N-methylpyridinium acetate) prodrug of paclitaxel induces superior antitumor responses in preclinical cancer models
Wrasidlo, W.; Gaedicke, G.; Guy, R. K.; Renaud, J.; Pitsinos, E. N.; Nicolaou, K. C.; Reisfeld, R. A.; Lode, H. N. Bioconjugate Chemistry 2002, 13, 1093–1099
- Synthetic studies towards trichodimerol and related vertinoid polyketides
Pitsinos, E.N.; Vidali, V.P.; Couladouros, E.A. ARKIVOC 2002, 13, 105–110
- Synthesis of o-brominated diaryl ethers using symmetrical iodonium salts:
Application to the synthesis of Bastadin precursors Couladouros, E.A.; Moutsos, V.I.; Pitsinos, E.N. ARKIVOC 2003, 15, 92–101
- Synthesis and evaluation of three novel scyphostatin analogues as neutral sphingomyelinase inhibitors
Pitsinos, E.N.; Wascholowski, V.; Karaliota, S.; Rigou, C.; Couladouros, E.A.; Giannis, A. ChemBioChem 2003, 4, 1223–1225
- Synthetic studies towards oxazinins. An expedient first total synthesis and proof of the absolute stereochemistry of oxazinin-3
Couladouros, E.A.; Moutsos, V.I.; Pitsinos, E.N. Tetrahedron Letters 2004, 45, 7779–7781
- A general method for the synthesis of bastaranes and isobastaranes. First total synthesis of bastadins 5, 10, 12, 16, 20 and 21
Couladouros, E.A.; Pitsinos, E.N.; Moutsos, V.I.; Sarakinos, G. Chemistry - A European Journal 2005, 11, 406–421
- Short and efficient route to the fully functionalized core of scyphostatin
Pitsinos, E.N.; Cruz, A. Organic Letters 2005, 7, 2245–2248
- Synthesis and biological evaluation of novel steroid-modified ether phospholipids
Karantonis, H.C.; Pitsinos, E.N.; Antonopoulou, S.; Couladouros, E.A.; Demopoulos, C.A. Chemistry and Physics of Lipids 2005, 138, 12–19
- Influence of the scyphostatin side-chain on the mode of inhibition of neutral sphingomyelinase
Wascholowski, V.; Giannis, A.; Pitsinos, E.N. ChemMedChem 2006, 1, 718–721
- Oxazinins from toxic mussels: isolation of a novel oxazinin and reassignment of the C-2 configuration of oxazinin-1 and -2 on the basis of synthetic models
Ciminiello, P.; Dell'Aversano, C.; Fattorusso, E.; Forino, M.; Magno, S.; Santelia, F.U.; Moutsos, V.I.; Pitsinos, E.N.; Couladouros, E.A. Tetrahedron 2006, 62, 7738–7743
- Synthesis of enantiopure (S)-7-hydroxy-3-amino-3,4-dihydro-2H-1-benzopyran en route to (+)-scyphostatin
Pitsinos, E.N.; Moutsos, V.I.; Vageli, O. Tetrahedron Letters 2007, 48, 1523–1526
- Synthetic bastadins modify the activity of ryanodine receptors in cultured cerebellar granule cells
Ziemińska, E.; Stafiej, A.; Pitsinos, E.N.; Couladouros, E.A.; Moutsos, V.; Kozłowska, H.; Toczyłowska, B.; Łazarewicz, J.W. NeuroSignals 2006-07, 15, 283–292
- Stereo-structural determination of three novel oxazinins isolated from Adriatic mussels via a synthetic and NMR-based approach
Ciminiello, P.; Dell’Aversano, C.; Fattorusso, E.; Forino, M.; Grauso, L.; Santelia, F.U.; Tartaglione, L.; Moutsos, V.I.; Pitsinos, E.N.; Couladouros, E.A. European Journal of Organic Chemistry 2007, 5434–5439
- Tumor necrosis factor-α promotes malignant pleural effusion
Stathopoulos, G.T.; Kollintza, A.; Moschos, A.; Psallidas, I.; Sherrill, T.P.; Pitsinos, E.N.; Vassiliou, S.; Karatza, M.; Papiris, S.A.; Graf, D.; Orphanidou, D.; Light, R.W.; Roussos, C.; Blackwell, T.S.; Kalomenidis, I. Cancer Research 2007, 67, 9825–9834
- Stereoselective syntheses of 2,6-disubstituted piperidin-3-oles (alkaloid lipids)
Koulocheri, S.D.; Pitsinos, E.N.; Haroutounian, S.A. Current Organic Chemistry 2008, 12, 1454–1467
- Open-chain half-bastadins mimic the effects of cyclic bastadins on calcium homeostasis in cultured neurons
Zieminska, E.; Lazarewicz, J.W.; Couladouros, E.A.; Moutsos,V.I.; Pitsinos, E.N. Bioorganic & Medicinal Chemistry Letters 2008, 18, 5734–5737
- Synthesis and characterization of novel natural product-Gd(III) MRI contrast agent conjugates
Efthimiadou, E.K.; Katsarou,M.E.; Fardis, M.; Zikos, C.; Pitsinos, E.N.; Kazantzis, A.; Leondiadis, L.; Sagnou, M.; Vourloumis, D. Bioorganic & Medicinal Chemistry Letters 2008, 18, 6058–6061
- Synthesis of novel laurenditerpenol analogues and their evaluation as HIF-1 activation inhibitors
Athinaios, N; Kazantzis, A.; Putzker, K.; Lewis, J.; Pitsinos, E.N. Letters in Organic Chemistry 2009, 6, 269–271
- Total synthesis of (+)-Scyphostatin featuring an enantioselective and highly efficient route to the side-chain via Zr-catalyzed asymmetric carboalumination of alkenes (ZACA)
Pitsinos, E.N.; Athinaios, N.; Xu, Z.; Wang, G.; Negishi, E.-I. Chemical Communications 2010, 46, 2200-2202
- Diaryl ether formation in the synthesis of natural products
Pitsinos, E.N.; Vidali, V.P.; Couladouros, E.A. European Journal of Organic Chemistry 2011, 1207-1222
- Enantioselective total synthesis of (–)-laurenditerpenol
Pitsinos, E.N.; Athinaios, N.; Vidali, V.P. Organic Letters 2012, 14, 4666-4669
- Bioefficacy of acyclic monoterpenes and their saturated derivatives against the West Nile vector Culex pipiens
Michaelakis, A.; Vidali, VP.; Papachristos, D.P.; Pitsinos, E.N.; Koliopoulos, G.; Couladouros, E.A; Polissiou, M.G.; Kimbaris, A.C. Chemosphere 2014, 96, 74–80.
- A fast entry to furanoditerpenoid-based Hedgehog signaling inhibitors: Identifying essential structural features
Chatzopoulou, M.; Antoniou, A.; Pitsinos, E.N.; Bantzi, M.; Koulocheri, S.D.; Haroutounian, S.A.; Giannis, A.G Organic Letters 2014, 16, 3344-3347.
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Last Updated on Friday, 26 September 2014 08:56 |
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